CP-724714 (b)

CAS No. 537705-08-1

CP-724714 (b)( —— )

Catalog No. M14915 CAS No. 537705-08-1

CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CP-724714 (b)
  • Note
    Research use only, not for human use.
  • Brief Description
    CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM.
  • Description
    CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc in cell-free assays. Phase 2.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    EGFR
  • Recptor
    HER2/ErbB2
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    537705-08-1
  • Formula Weight
    469.53
  • Molecular Formula
    C27H27N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    N/A
  • SMILES
    CCOC(=O)NC/C=C/C1=CC2=C(C=C1)N=CN=C2NC3=CC(=C(C=C3)OC4=CN=C(C=C4)C)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1 Jani JP, et al. Cancer Res, 2007, 67(20), 9887-9893. 2 Feng B, et al. Toxicol Sci, 2009, 108(2), 492-500.
molnova catalog
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